Bretazenil CAS: 84379-13-5

CAS NO: 84379-13-5
Our products are for scientific research use only

chemical name : Bretazenil
Molecular Formula :C19H20BrN3O3
Synonyms :Ro 16-6028
benzodiazepine-1-carboxylic acid, 1,1-dimethylethyl ester
CAS :84379-13-5
Description Review
Description
Our products are for scientific research use only

Benefits of Bretazenil for Health
Bretazenil, a benzodiazepine analog, is mainly used to treat anxiety and seizures. It is recognized for its milder sedative effect in comparison to other benzodiazepines, rendering it a more suitable choice for patients who require anxiety management without requiring substantial sedation.



Possible Consequences
Anxiolytic: lowers stress and anxiety
Medications used to treat or prevent epileptic seizures are known as anticonvulsants.
The sedative effect is less intense than that of other benzodiazepines, but it is nevertheless effective in reducing agitation and inducing calm.
Relieves muscular spasms
Product Mechanism
Bretazenil acts on the brain's gamma-aminobutyric acid (GABA) receptors by modifying their activation. Bretazenil's calming, anticonvulsant, and muscle-relaxant characteristics are due to its ability to enhance the impact of GABA, an inhibitory neurotransmitter.

What are the risks and effects?
Safety Profile
The partial agonist action of bretazenil at GABA receptors contributes to its positive safety profile. Some complete agonists, such as diazepam and alprazolam, are associated with a greater number of adverse effects than partial agonism.






Bretazenil CAS: 84379-13-5
Side Effects
Drowsiness
Dizziness
Fatigue
Nausea
Headache
Rare yet serious adverse effects might consist of:

Respiratory depression.
Prolonged use induces dependence.
Having trouble thinking

Dosage Information: The amount of Bretazenil a person takes should depend on their needs and how well they respond to treatment. It is common practice to start with smaller dosages and gradually increase or decrease them as needed. Because of the pharmacological features it has, it is highly recommended to adhere to the instructions provided by a healthcare practitioner.

Contraindications
Bretazenil is contraindicated in certain individuals:

Severe respiratory insufficiency
In summary



Bretazenil is a versatile benzodiazepine analog with a unique profile that offers anxiolytic, anticonvulsant, and muscle-relaxant benefits with a reduced sedative impact. Its partial agonist action has the benefit of reducing side effects and dependence hazards, making it an attractive alternative in clinical practice. But it's important to think carefully about doses, safety, and situations where it shouldn't be used.

People Also Ask


What is the purpose of Bretazenil?
The anticonvulsant and anxiolytic effects of bretazenil make it a popular medicine. With less sedation than other benzodiazepines, it treats anxiety and epilepsy.

In what ways is Bretazenil similar to Diazepam?
Bretazenil has a gentler sedative effect and is less likely to cause dependence than diazepam. It functions as a partial agonist at GABA receptors, whereas diazepam is a full agonist, resulting in more potent sedative and muscle relaxant effects.

Is it safe to take Bretazenil for a long time?
The partial agonist action of bretazenil makes it a more benign long-term benzodiazepine option. On the other hand, prolonged usage should still be supervised by a medical practitioner in order to avoid the possibility of developing a dependence and experiencing adverse consequences.

Is Bretazenil addictive?
Bretazenil has a lesser dependence risk than full-agonist benzodiazepines, although chronic usage may lead to addiction. It is imperative that this drug be used under close physician supervision.

What should I do if I miss a dosage of Bretazenil?
Take your Bretazenil as soon as you remember if you forget to. If your next dosage is nearly here, skip the missed one and go back to your usual dosing plan. Do not duplicate the dosage to make up for a missing one. Always adhere to your healthcare provider's directions.





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Some common synonyms for Bretazenil include Ro11-6896, MK-0677, L-79206, and 7-(2,2-Diphenyl-1-oxoethyl)-6-(3-propenyl)-4H,5H,6H,7H,8H-Imidazo[1,5-a][1,4]benzodiazepine-3-carboxylic acid methyl ester.

Similar Competitive Products

  • Diazepam
  • Clonazepam
  • Lorazepam
  • Alprazolam
  • Etizolam
  • Diazepam: Widely used for anxiety, muscle spasms, and seizures.
  • Alprazolam: Commonly prescribed for anxiety and panic disorders.
  • Lorazepam: Utilized for its anxiolytic, sedative, and anticonvulsant properties.
  • Clonazepam: Known for treating panic disorders and seizure conditions.
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